SCHEMBL4554534

SCHEMBL4554534

CC(C)CC1c2ccc(NC(=O)C(=S)NN)cc2CCN1C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 11/20 0.40
MTNR1A P48039 2/20 0.37
HHAT Q5VTY9 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
CYP2D6 P10635 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4554899 0.83 MTNR1B (0.38) MTNR1BMTNR1AMEN1KMT2A
SCHEMBL4555618 0.82 MTNR1B (0.42) MTNR1BMTNR1AMEN1KMT2A
SCHEMBL4554533 0.81 DPP4 (0.35) KMT2APOLB
SCHEMBL3664253 0.78 MTNR1B (0.47) MTNR1BMTNR1AHHAT
SCHEMBL3665398 0.77 ROCK2 (0.44) MTNR1BMTNR1A
SCHEMBL4032581 0.76 MTNR1B (0.48) MTNR1BMTNR1A
SCHEMBL2123940 0.75 MTNR1B (0.47) MTNR1BMTNR1AMEN1KMT2A
SCHEMBL4555438 0.73 MTNR1B (0.38) MTNR1BMTNR1A
SCHEMBL2123210 0.73 MTNR1B (0.45) MTNR1BMTNR1A
SCHEMBL2123219 0.72 MTNR1B (0.43) MTNR1BMTNR1AHHAT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125799-A1 THIADIAZOLE DERIVATIVES, INHIBITORS OF STEAROYL-COA DESATURASE Smithkline Beecham Corporation (US) 2009-12-02 EP disclosed
WO-2008104524-A1 THIADIAZOLE DERIVATIVES, INHIBITORS OF STEAROYL-COA DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2008-09-04 WO disclosed