SCHEMBL4554899

SCHEMBL4554899

CC(C)CC1c2ccc(NC(=O)C(=S)N3CCOCC3)cc2CCN1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 4/20 0.38
ALDH1A1 P00352 4/20 0.37
MAPT P10636 3/20 0.37
LMNA P02545 2/20 0.37
KDM4E B2RXH2 2/20 0.37
DUSP3 P51452 1/20 0.37
PTPN5 P54829 1/20 0.37
PTPN11 Q06124 1/20 0.37
APOBEC3G Q9HC16 1/20 0.37
MAPK1 P28482 1/20 0.37
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
RAB9A P51151 4/20 0.36
HTT P42858 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HPGD P15428 1/20 0.36
ALOX15 P16050 1/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4554534 0.83 MTNR1B (0.40) MTNR1BMEN1KMT2AMTNR1A
SCHEMBL4554898 0.82 LMNA (0.39) ALDH1A1MAPTLMNAKDM4EDUSP3
SCHEMBL4555618 0.79 MTNR1B (0.42) MTNR1BALDH1A1MAPTLMNAKDM4E
SCHEMBL3665398 0.74 ROCK2 (0.44) MTNR1BALDH1A1LMNAMTNR1A
SCHEMBL4032581 0.73 MTNR1B (0.48) MTNR1BMTNR1A
SCHEMBL13347343 0.73 LMNA (0.50) ALDH1A1MAPTLMNAKDM4EDUSP3
SCHEMBL2123940 0.72 MTNR1B (0.47) MTNR1BLMNAMEN1KMT2AMTNR1A
SCHEMBL3664253 0.72 MTNR1B (0.47) MTNR1BMTNR1A
SCHEMBL4555438 0.71 MTNR1B (0.38) MTNR1BMTNR1A
SCHEMBL2123210 0.70 MTNR1B (0.45) MTNR1BMTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125799-A1 THIADIAZOLE DERIVATIVES, INHIBITORS OF STEAROYL-COA DESATURASE Smithkline Beecham Corporation (US) 2009-12-02 EP disclosed
WO-2008104524-A1 THIADIAZOLE DERIVATIVES, INHIBITORS OF STEAROYL-COA DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2008-09-04 WO disclosed