SCHEMBL4554910

SCHEMBL4554910

CN(C(=O)c1ccc2c(c1)CCN(C(=O)O)C2C(C)(C)C)c1nnc(COc2ccccc2Cl)s1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 6/20 0.35
SMN1; SMN2 Q16637 5/20 0.35
NPC1 O15118 4/20 0.35
RAB9A P51151 4/20 0.35
HTT P42858 3/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPT P10636 1/20 0.35
MDM2 Q00987 1/20 0.35
GPR55 Q9Y2T6 1/20 0.35
MEN1 O00255 4/20 0.33
KMT2A Q03164 4/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TP53 P04637 2/20 0.33
MITF O75030 1/20 0.33
XBP1 P17861 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4554911 0.88 MTNR1B (0.36) HPGDSMN1; SMN2NPC1RAB9AHTT
SCHEMBL4555464 0.84 LMNA (0.47) HPGDSMN1; SMN2NPC1RAB9AHTT
SCHEMBL4554891 0.81 FFAR1 (0.44)
SCHEMBL3729629 0.79 ESR2 (0.47) SMN1; SMN2NPC1RAB9AHTTL3MBTL1
SCHEMBL3723598 0.76 SYK (0.41) HPGDSMN1; SMN2NPC1RAB9AHTT
Hydrochloric Acid SCHEMBL3729480 0.76 SYK (0.41) HPGDSMN1; SMN2NPC1RAB9AHTT
SCHEMBL4553190 0.73 LMNA (0.46) HPGDSMN1; SMN2HTTALDH1A1MAPT
SCHEMBL4555465 0.72 LMNA (0.44) HPGDSMN1; SMN2HTTALDH1A1MEN1
SCHEMBL4554892 0.69 FFAR1 (0.43)
SCHEMBL4032578 0.67 ESR1 (0.51) GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125799-A1 THIADIAZOLE DERIVATIVES, INHIBITORS OF STEAROYL-COA DESATURASE Smithkline Beecham Corporation (US) 2009-12-02 EP disclosed
WO-2008104524-A1 THIADIAZOLE DERIVATIVES, INHIBITORS OF STEAROYL-COA DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2008-09-04 WO disclosed