SCHEMBL4555401

SCHEMBL4555401

Cc1ccc(-c2c(C(N)=O)cccc2C(F)(F)F)c(N)c1-c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FABP4 P15090 2/20 0.46
SCN9A Q15858 6/20 0.40
BCAT2 O15382 1/20 0.40
PARP1 P09874 1/20 0.40
NR1H2 P55055 1/20 0.40
NR1H3 Q13133 1/20 0.40
PDK2 Q15119 1/20 0.40
TAS2R14 Q9NYV8 2/20 0.39
RORC P51449 1/20 0.38
MYC P01106 1/20 0.38
CYP3A4 P08684 1/20 0.37
CD38 P28907 1/20 0.37
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
AURKA O14965 1/20 0.36
RPS6KB1 P23443 1/20 0.36
AURKB Q96GD4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28812647 0.84 FABP4 (0.57) FABP4SCN9ABCAT2PARP1NR1H2
SCHEMBL530568 0.83 FABP4 (0.58) FABP4SCN9ABCAT2PARP1NR1H2
SCHEMBL30339795 0.83 FABP4 (0.58) FABP4SCN9ABCAT2PARP1NR1H2
SCHEMBL29286691 0.77 PARP1 (0.40) FABP4SCN9APARP1PDK2CYP3A4
SCHEMBL6173681 0.76 PARP1 (0.52) SCN9ABCAT2PARP1PDK2TAS2R14
SCHEMBL30241242 0.76 FABP4 (0.45) FABP4SCN9APARP1NR1H2NR1H3
SCHEMBL4555403 0.75 BRD4 (0.41) FABP4SCN9APARP1PDK2MYC
SCHEMBL4776531 0.74 FABP4 (0.46) FABP4SCN9ABCAT2PARP1NR1H2
SCHEMBL7161543 0.74 BCAT2 (0.51) FABP4SCN9ABCAT2PARP1NR1H2
SCHEMBL27475690 0.74 BCAT2 (0.47) FABP4BCAT2MYC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121692-A1 SUBSTITUTED HETEROCYCLES AS JANUS KINASE INHIBITORS Incyte Corporation (US) 2009-11-25 EP disclosed
WO-2008079965-A1 SUBSTITUTED HETEROCYCLES AS JANUS KINASE INHIBITORS INCYTE CORPORATION (US) 2008-07-03 WO disclosed