SCHEMBL4555607

SCHEMBL4555607

NC(=O)c1ccc2c(c1)CCNC2c1nccs1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NNMT P40261 2/20 0.41
HTR2C P28335 1/20 0.39
MAPKAPK2 P49137 1/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
HSD11B1 P28845 1/20 0.35
CHEK2 O96017 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
KDM1A O60341 2/20 0.34
HTR1D P28221 5/20 0.34
HTR1B P28222 2/20 0.34
DRD2 P14416 3/20 0.33
HTR2A P28223 3/20 0.33
HTR1A P08908 2/20 0.33
CTSA P10619 1/20 0.33
DRD4 P21917 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29830988 0.76 HTR2C (0.37) HTR2CHSD11B1HTR1A
SCHEMBL29831263 0.75 RECQL (0.55) HTR2CMEN1KMT2A
SCHEMBL4555606 0.75 CHEK2 (0.36) NNMTHTR2CCHEK2MEN1KMT2A
SCHEMBL4701188 0.74 CHEK2 (0.35) NNMTCHEK2MEN1KMT2AKDM1A
SCHEMBL26101504 0.73 NNMT (0.44) NNMTMAPKAPK2CA1CA2CA7
Hydrochloric Acid SCHEMBL4875139 0.72 MEN1 (0.37) NNMTMAPKAPK2CA1CA2CA7
SCHEMBL20504221 0.70 PRCP (0.53) NNMTMAPKAPK2MEN1KMT2AKDM1A
SCHEMBL20504355 0.70 MAPKAPK2 (0.44) NNMTMAPKAPK2MEN1KMT2AKDM1A
SCHEMBL13728706 0.69 AKR1C3 (0.39) HSD11B1DRD4
SCHEMBL23304573 0.68 OPRM1 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103998027-A Methods of using SCD1 antagonists for cancer therapy HOFFMANN LA ROCHE 2014-08-20 CN disclosed
EP-2125799-A1 THIADIAZOLE DERIVATIVES, INHIBITORS OF STEAROYL-COA DESATURASE Smithkline Beecham Corporation (US) 2009-12-02 EP disclosed
WO-2008104524-A1 THIADIAZOLE DERIVATIVES, INHIBITORS OF STEAROYL-COA DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2008-09-04 WO disclosed