SCHEMBL4555853

SCHEMBL4555853

Cc1cccc2[nH]c(C(F)(F)C3(C(=O)N[C@@H](CP(=O)(O)O)C(=O)O)Nc4ccccc4N3C)nc12

nearest known ligand 0.32

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
F9 P00740 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
MMP2 P08253 2/20 0.31
MMP9 P14780 2/20 0.31
MMP8 P22894 2/20 0.31
KDM4E B2RXH2 1/20 0.31
HPGD P15428 1/20 0.31
HCRTR1 O43613 1/20 0.30
HCRTR2 O43614 1/20 0.30
HRH4 Q9H3N8 1/20 0.30
MMP13 P45452 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2524929 0.70 TPSAB1 (0.51)
SCHEMBL2526178 0.64 PIN1 (0.41) ALDH1A1
SCHEMBL2526173 0.64 PIN1 (0.41) ALDH1A1
SCHEMBL6830451 0.58 PIN1 (0.49)
SCHEMBL8598047 0.58 GAA (0.63) ALDH1A1TDP1KDM4EHPGD
Trifluoroacetic Acid SCHEMBL6951531 0.56 ALDH1A1 (0.47) ALDH1A1TDP1MMP2MMP9MMP8
Phosphoric Acid SCHEMBL11576943 0.56 MAOB (0.51) ALDH1A1TDP1MMP2MMP9MMP8
SCHEMBL11001624 0.55 ALDH1A1 (0.53) ALDH1A1TDP1MMP2MMP9MMP8
SCHEMBL6759197 0.55 MGAM (0.50) ALDH1A1TDP1
SCHEMBL4352212 0.55 MGAM (0.55) ALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125753-A1 FUSED HETEROCYCLIC COMPOUNDS HAVING CRF ANTAGONISTIC ACTIVITY Takeda Pharmaceutical Company Limited (JP) 2009-12-02 EP claimed
WO-2008082003-A1 FUSED HETEROCYCLIC COMPOUNDS HAVING CRF ANTAGONISTIC ACTIVITY TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-07-10 WO claimed