SCHEMBL4556755

SCHEMBL4556755

Cc1nnc(-c2ccc(N3CCC4(CCc5c(Cl)ccc(Cl)c5O4)CC3)nc2)o1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 5/20 0.39
SCD O00767 9/20 0.39
HRH3 Q9Y5N1 1/20 0.37
TTK P33981 1/20 0.36
ATR Q13535 1/20 0.35
WNT1 P04628 1/20 0.34
GSK3B P49841 1/20 0.34
DYRK1A Q13627 1/20 0.34
PCSK9 Q8NBP7 1/20 0.34
DGAT1 O75907 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4555897 0.87 CNR2 (0.42) CNR2SCDHRH3TTKATR
SCHEMBL8192205 0.74 CNR2 (0.50) CNR2HRH3ATR
SCHEMBL4557053 0.71 HDAC1 (0.47) SCDCYP3A4
SCHEMBL4556849 0.68 SCD (0.48) SCD
SCHEMBL4557042 0.66 CNR2 (0.39) CNR2DGAT1CYP2C9
SCHEMBL1435967 0.64 NPC1 (0.65) PCSK9
SCHEMBL13930462 0.63 SCD (0.53) SCD
SCHEMBL11884342 0.62 NOTUM (0.60) CYP1A2CYP2C19
SCHEMBL4259675 0.61 SCD (0.53) SCDCYP3A4CYP2D6
SCHEMBL1589838 0.60 SCD (0.48) CNR2SCDCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009037542-A2 SPIROCYCLIC COMPOUNDS AS STEAROYL COA DESATURASE INHIBITORS GLENMARK PHARMACEUTICALS, S.A. (US) 2009-03-26 WO disclosed
WO-2009037542-A2 SPIROCYCLIC COMPOUNDS AS STEAROYL COA DESATURASE INHIBITORS GLENMARK PHARMACEUTICALS, S.A. (US) 2009-03-26 WO disclosed