SCHEMBL4557042

SCHEMBL4557042

Clc1cccc2c1OC1(CC2)CCN(c2ccc(-c3nnn[nH]3)cn2)CC1

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 8/20 0.39
CNR1 P21554 1/20 0.38
TRPM8 Q7Z2W7 7/20 0.38
DGAT1 O75907 4/20 0.38
TNKS O95271 1/20 0.36
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4555897 0.79 CNR2 (0.42) CNR2CNR1TRPM8DGAT1
SCHEMBL4445219 0.73 TRPM8 (0.44) CNR2TRPM8
SCHEMBL4450951 0.71 SCD (0.53) CNR2TRPM8CYP2C9
SCHEMBL13930227 0.70 TRPM8 (0.39) CNR2CNR1TRPM8
SCHEMBL4556505 0.69 TRPM8 (0.43) TRPM8
SCHEMBL4556755 0.66 CNR2 (0.39) CNR2DGAT1CYP2C9
SCHEMBL16496070 0.65 SCD (0.58)
SCHEMBL13770570 0.64 TRPM8 (0.49) TRPM8
SCHEMBL4556993 0.64 HDAC6 (0.50)
SCHEMBL4443503 0.63 DRD2 (0.43) TRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009037542-A2 SPIROCYCLIC COMPOUNDS AS STEAROYL COA DESATURASE INHIBITORS GLENMARK PHARMACEUTICALS, S.A. (US) 2009-03-26 WO claimed
WO-2009037542-A2 SPIROCYCLIC COMPOUNDS AS STEAROYL COA DESATURASE INHIBITORS GLENMARK PHARMACEUTICALS, S.A. (US) 2009-03-26 WO disclosed