SCHEMBL455841

SCHEMBL455841

NC(=O)c1ccc(C2(c3cnc4c(NCCS(N)(=O)=O)cc(Cl)nn34)CC2)cc1

nearest known ligand 0.31

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
PIK3CD O00329 1/20 0.31
PIK3R1 P27986 1/20 0.31
PIK3CA P42336 1/20 0.31
PIK3CB P42338 1/20 0.31
PIK3CG P48736 1/20 0.31
HSD11B1 P28845 1/20 0.31
PI4KB Q9UBF8 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL457969 0.76 TTK (0.45)
SCHEMBL456964 0.74 TTK (0.36) ERN1
SCHEMBL456370 0.72 TTK (0.41) PI4KB
SCHEMBL455843 0.70 ERN1 (0.46) ERN1
SCHEMBL10279180 0.64 TTK (0.56) ERN1
SCHEMBL470191 0.62 FYN (0.47) ERN1
SCHEMBL12466787 0.61 ERN1 (0.39) ERN1
SCHEMBL18208715 0.57 TTK (0.36) ERN1
SCHEMBL10383734 0.56 ADRB3 (0.38) ERN1
SCHEMBL10382989 0.54 ALDH1A1 (0.39) TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614063-A1 SUBSTITUTED IMIDAZOPYRIDAZINES Bayer Intellectual Property GmbH (DE) 2013-07-17 EP disclosed
WO-2012032031-A1 SUBSTITUTED IMIDAZOPYRIDAZINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-03-15 WO disclosed