SCHEMBL4563606

SCHEMBL4563606

C=CCc1nccn1-c1cccc2ccccc12

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.42
MAPK1 P28482 1/20 0.42
PI4KA P42356 1/20 0.37
PI4K2B Q8TCG2 1/20 0.37
PI4K2A Q9BTU6 1/20 0.37
PI4KB Q9UBF8 1/20 0.37
HCAR1 Q9BXC0 1/20 0.37
ALDH1A1 P00352 3/20 0.35
TP53 P04637 1/20 0.34
NOTUM Q6P988 1/20 0.34
KMT2A Q03164 1/20 0.34
HPGD P15428 2/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34
GFER P55789 1/20 0.34
ADRB2 P07550 1/20 0.33
POLB P06746 1/20 0.33
P2RX4 Q99571 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8564307 0.77 NPC1 (0.42) NPC1MAPK1PI4KAPI4K2BPI4K2A
SCHEMBL9397982 0.75 CYP3A4 (0.43) NPC1ALDH1A1KMT2AGAAPOLB
SCHEMBL5638922 0.72 NPC1 (0.49) NPC1MAPK1PI4KAPI4K2BPI4K2A
SCHEMBL28330184 0.72 PI4KA (0.49) NPC1MAPK1PI4KAPI4K2BPI4K2A
SCHEMBL9405397 0.72 NPC1 (0.49) NPC1MAPK1PI4KAPI4K2BPI4K2A
SCHEMBL28367072 0.72 NPC1 (0.45) NPC1MAPK1PI4KAPI4K2BPI4K2A
SCHEMBL27659057 0.70 P2RX4 (0.46) NPC1MAPK1PI4KAPI4K2BPI4K2A
SCHEMBL4866386 0.70 NPC1 (0.46) NPC1MAPK1PI4KAPI4K2BPI4K2A
SCHEMBL11345662 0.69 TDP1 (0.42) HCAR1ALDH1A1HPGDLMNAGAA
SCHEMBL27944468 0.69 NPC1 (0.45) NPC1MAPK1PI4KAPI4K2BPI4K2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061464-A2 COMBINATION THERAPY FOR TUMORAL DISEASE TREATMENT Ramot, at Tel Aviv University Ltd. (IL) 2009-05-27 EP disclosed
WO-2008032324-A2 COMBINATION THERAPY FOR TUMORAL DISEASE TREATMENT RAMOT AT TEL AVIV UNIVERSITY LTD. (IL) 2008-03-20 WO disclosed