SCHEMBL8564307

SCHEMBL8564307

CC(C)Cc1nccn1-c1cccc2ccccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.42
MAPK1 P28482 1/20 0.42
CNR2 P34972 1/20 0.41
KMT2A Q03164 1/20 0.39
PI4KA P42356 1/20 0.37
PI4K2B Q8TCG2 1/20 0.37
PI4K2A Q9BTU6 1/20 0.37
PI4KB Q9UBF8 1/20 0.37
HCAR1 Q9BXC0 1/20 0.37
TP53 P04637 1/20 0.36
ELANE P08246 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
TSHR P16473 1/20 0.35
DRD1 P21728 1/20 0.35
DRD5 P21918 1/20 0.35
ALDH1A1 P00352 1/20 0.35
P2RX4 Q99571 1/20 0.35
NOTUM Q6P988 1/20 0.34
TLR8 Q9NR97 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4563606 0.77 NPC1 (0.42) NPC1MAPK1KMT2API4KAPI4K2B
SCHEMBL9405397 0.75 NPC1 (0.49) NPC1MAPK1KMT2API4KAPI4K2B
SCHEMBL20402553 0.75 HTR1A (0.34)
SCHEMBL5638922 0.72 NPC1 (0.49) NPC1MAPK1KMT2API4KAPI4K2B
SCHEMBL28330184 0.72 PI4KA (0.49) NPC1MAPK1KMT2API4KAPI4K2B
SCHEMBL31202561 0.71 CYP2A6 (0.46) NPC1MAPK1PI4KAPI4K2BPI4K2A
SCHEMBL27659057 0.70 P2RX4 (0.46) NPC1MAPK1PI4KAPI4K2BPI4K2A
SCHEMBL4866386 0.70 NPC1 (0.46) NPC1MAPK1PI4KAPI4K2BPI4K2A
SCHEMBL28367072 0.69 NPC1 (0.45) NPC1MAPK1KMT2API4KAPI4K2B
SCHEMBL27944468 0.69 NPC1 (0.45) NPC1MAPK1KMT2API4KAPI4K2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821675-A1 NOVEL HYDROXAMIC ACID AND AMINO-CARBOXYLATE COMPOUNDS AS METALLOPROTEASE AND TNF INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-02-04 EP disclosed
WO-1996033176-A1 NOVEL HYDROXAMIC ACID AND AMINO-CARBOXYLATE COMPOUNDS AS METALLOPROTEASE AND TNF INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-10-24 WO disclosed