SCHEMBL4564236

SCHEMBL4564236

CC1NCc2cc(OC(=O)O)ccc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 4/20 0.37
ACHE P22303 5/20 0.36
OPRD1 P41143 2/20 0.33
KDM4E B2RXH2 2/20 0.33
LMNA P02545 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
OPRK1 P41145 1/20 0.33
ESR1 P03372 1/20 0.33
PGR P06401 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
AR P10275 1/20 0.33
CHRM1 P11229 1/20 0.33
TBXA2R P21731 1/20 0.33
ADRA1A P35348 1/20 0.33
SLC6A3 Q01959 1/20 0.33
ATM Q13315 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HTR2C P28335 1/20 0.33
CYP3A4 P08684 2/20 0.33
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4404012 0.79 HTR2C (0.50) OPRM1HTR2C
Hydrochloric Acid SCHEMBL30931423 0.71 ACHE (0.43) OPRM1ACHELMNASMN1; SMN2ESR1
SCHEMBL4563940 0.70 ITGB3 (0.38) KDM4ESMN1; SMN2
SCHEMBL13460942 0.70 CHRNB2 (0.39) ACHEKDM4ESLC6A3HTR2C
SCHEMBL18664431 0.70 CHRNB2 (0.39) ACHEKDM4ESLC6A3HTR2C
Hydrochloric Acid SCHEMBL7278190 0.69 ITGB3 (0.40) KDM4ESMN1; SMN2
SCHEMBL2898828 0.68 PNMT (0.56) HTR2C
SCHEMBL6671284 0.68 PNMT (0.56) HTR2C
SCHEMBL29396876 0.68 PNMT (0.56) HTR2C
Hydrochloric Acid SCHEMBL2895888 0.67 PNMT (0.54) HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2132193-A1 SUBSTITUTED PYRROLIDINE AMIDES, THE PRODUCTION THEREOF, AND THE USE THEREOF AS MEDICATIONS Boehringer Ingelheim International GmbH (DE) 2009-12-16 EP disclosed
WO-2008116881-A1 SUBSTITUTED PYRROLIDINE AMIDES, THE PRODUCTION THEREOF, AND THE USE THEREOF AS MEDICATIONS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-10-02 WO disclosed