SCHEMBL4565641

SCHEMBL4565641

COC(=O)Cc1c(C)n(Cc2ccc(Cl)cc2)c2cc(Cl)c(C)cc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.58
CYP1A2 P05177 2/20 0.58
CYP3A4 P08684 2/20 0.58
CYP2C9 P11712 2/20 0.58
TSHR P16473 2/20 0.58
CYP2C19 P33261 2/20 0.58
PMP22 Q01453 2/20 0.58
MEN1 O00255 1/20 0.58
RGS12 O14924 1/20 0.58
ALDH1A1 P00352 1/20 0.58
MAPT P10636 1/20 0.58
PKM P14618 1/20 0.58
NFKB1 P19838 1/20 0.58
MAPK1 P28482 1/20 0.58
GNAI1 P63096 1/20 0.58
KMT2A Q03164 1/20 0.58
HIF1A Q16665 1/20 0.58
PLA2G2A P14555 10/20 0.57
PTGS2 P35354 5/20 0.51
CNR2 P34972 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3003631 0.87 LMNA (0.68) LMNACYP1A2CYP3A4CYP2C9TSHR
SCHEMBL14106891 0.87 PLA2G2A (0.50) LMNACYP1A2CYP3A4CYP2C9TSHR
SCHEMBL8292638 0.85 MAPT (0.63) LMNACYP1A2CYP3A4CYP2C9TSHR
SCHEMBL12571243 0.81 LMNA (0.56) LMNACYP1A2CYP3A4CYP2C9TSHR
SCHEMBL8292072 0.81 PLA2G2A (0.61) LMNACYP1A2CYP3A4CYP2C9TSHR
SCHEMBL2003800 0.80 LMNA (0.71) LMNACYP1A2CYP3A4CYP2C9TSHR
SCHEMBL5439155 0.78 LMNA (0.65) LMNACYP1A2CYP3A4CYP2C9TSHR
SCHEMBL2003118 0.77 LMNA (0.56) LMNACYP1A2CYP3A4CYP2C9TSHR
SCHEMBL2005651 0.77 LMNA (0.64) LMNACYP1A2CYP3A4CYP2C9TSHR
SCHEMBL3006501 0.76 PTGDR2 (0.64) LMNACYP1A2CYP3A4CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049520-A2 INDOLE COMPOUNDS Ironwood Pharmaceuticals, Inc. (US) 2009-04-22 EP disclosed
WO-2008019357-A2 INDOLE COMPOUNDS IRONWOOD PHARMACEUTICALS, INC. (US) 2008-02-14 WO disclosed