SCHEMBL4565736

SCHEMBL4565736

CC(C)(C)OC(=O)Nc1cccc(-n2cc(C(=O)O)cn2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.56
NFE2L2 Q16236 1/20 0.56
HPGDS O60760 1/20 0.52
ALKBH2 Q6NS38 1/20 0.52
P2RY14 Q15391 1/20 0.46
CYP17A1 P05093 1/20 0.46
XDH P47989 1/20 0.44
HDAC3 O15379 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
NAMPT P43490 1/20 0.43
EGLN1 Q9GZT9 1/20 0.42
ALKBH1 Q13686 1/20 0.42
MAPK13 O15264 1/20 0.41
MAPK8 P45983 1/20 0.41
MAPK12 P53778 1/20 0.41
MAPK10 P53779 1/20 0.41
MAPK11 Q15759 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6963518 0.79 SCD (0.48) HPGDSALKBH2HDAC3HDAC8NAMPT
SCHEMBL19252949 0.79 SCD (0.55) CYP17A1HDAC3HDAC1HDAC2HDAC8
SCHEMBL18704475 0.78 CYP17A1 (0.42) CYP17A1HDAC3HDAC1HDAC2HDAC8
SCHEMBL29435026 0.77 HDAC3 (0.58) CYP17A1HDAC3HDAC1HDAC2HDAC8
SCHEMBL222876 0.77 HDAC3 (0.58) CYP17A1HDAC3HDAC1HDAC2HDAC8
SCHEMBL22570944 0.76 NOTUM (0.50) KEAP1CYP17A1HDAC3HDAC1HDAC2
SCHEMBL7439456 0.76 HDAC3 (0.57) CYP17A1HDAC3HDAC1HDAC2HDAC8
SCHEMBL3510402 0.74 CYP17A1 (0.67) CYP17A1HDAC3HDAC1HDAC2HDAC8
SCHEMBL6165168 0.74 HPGDS (0.61) KEAP1NFE2L2HPGDSALKBH2EGLN1
SCHEMBL29029431 0.74 HDAC3 (0.56) CYP17A1HDAC3HDAC1HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044055-A2 AMIDE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-04-08 EP disclosed
WO-2008011131-A2 AMIDE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-01-24 WO disclosed