SCHEMBL4566586

SCHEMBL4566586

C=CCC1CNc2ccccc2O1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CASR P41180 1/20 0.44
HTR1A P08908 3/20 0.43
NISCH Q9Y2I1 1/20 0.42
HPGD P15428 2/20 0.41
HRH3 Q9Y5N1 1/20 0.37
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HSD17B10 Q99714 1/20 0.35
GAA P10253 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
BRD4 O60885 1/20 0.33
CREBBP Q92793 1/20 0.33
ALOX5 P09917 1/20 0.33
PARP1 P09874 1/20 0.33
NR3C1 P04150 1/20 0.32
PGR P06401 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8569387 0.81 ALDH1A1 (0.42) CASRHTR1ANISCHHPGDHRH3
SCHEMBL8569392 0.81 ALDH1A1 (0.42) CASRHTR1ANISCHHPGDHRH3
SCHEMBL8569391 0.81 ALDH1A1 (0.42) CASRHTR1ANISCHHPGDHRH3
SCHEMBL2638179 0.78 CASR (0.47) CASRHTR1ANISCHHPGDUSP2
SCHEMBL17150937 0.78 CASR (0.50) CASRHTR1ANISCHHPGDGAA
SCHEMBL8570483 0.78 CASR (0.47) CASRHTR1ANISCHHPGDUSP2
SCHEMBL3969657 0.78 CASR (0.47) CASRHTR1ANISCHHPGDUSP2
SCHEMBL3969660 0.78 CASR (0.47) CASRHTR1ANISCHHPGDUSP2
SCHEMBL30112409 0.78 CASR (0.50) CASRHTR1ANISCHHPGDGAA
SCHEMBL4824743 0.75 HPGD (0.51) CASRHTR1ANISCHHPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0304684-A1 Process for the preparation of benzoxazine derivatives DAIICHI SEIYAKU CO., LTD. (JP) 1989-03-01 EP claimed
WO-2009148659-A2 ANTIMALARIAL QUINOLINES AND METHODS OF USE THEREOF GEORGETOWN UNIVERSITY (US) 2009-12-10 WO disclosed