SCHEMBL4566627

SCHEMBL4566627

CN(C(=O)OCc1cn(S(=O)(=O)c2cccnc2)c(-c2cccnc2F)c1F)C(C)(C)C

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 1/20 0.33
ABCC8 Q09428 1/20 0.33
KCNJ11 Q14654 1/20 0.33
KCNJ8 Q15842 1/20 0.33
HTR6 P50406 1/20 0.33
CHRNB4 P30926 2/20 0.31
CHRNA3 P32297 2/20 0.31
NAMPT P43490 3/20 0.31
GAA P10253 2/20 0.31
GPBAR1 Q8TDU6 1/20 0.31
RORC P51449 1/20 0.31
TSHR P16473 1/20 0.31
GFER P55789 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
KAT5 Q92993 1/20 0.31
KAT8 Q9H7Z6 1/20 0.31
CHRNB2 P17787 1/20 0.30
CHRNA4 P43681 1/20 0.30
IDE P14735 1/20 0.30
KEAP1 Q14145 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4566745 0.86 TSHR (0.32) ABCC9ABCC8KCNJ11KCNJ8TSHR
SCHEMBL4566599 0.85 RXFP1 (0.35) HTR6GPBAR1SMN1; SMN2RXFP1
SCHEMBL4566561 0.85 HTR6 (0.40) HTR6RORCKEAP1
SCHEMBL2411042 0.83 HTR6 (0.33) ABCC9ABCC8KCNJ11KCNJ8HTR6
SCHEMBL4569945 0.83 ALDH1A1 (0.36) RORCKDM4E
SCHEMBL4566724 0.82
SCHEMBL2410178 0.82 NAMPT (0.37) NAMPTSMN1; SMN2
SCHEMBL4566781 0.81
SCHEMBL2413180 0.81 HTR6 (0.37) HTR6CHRNB4CHRNA3NAMPTGAA
SCHEMBL4566448 0.80 HTT (0.34) GAARXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed