SCHEMBL4569945

SCHEMBL4569945

CN(C(=O)OCc1cn(S(=O)(=O)c2ccccc2C#N)c(-c2cccnc2F)c1F)C(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 2/20 0.36
KDM2B Q8NHM5 1/20 0.33
NR1H3 Q13133 1/20 0.32
HTT P42858 1/20 0.31
HSD11B1 P28845 1/20 0.31
AOC3 Q16853 3/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
RORC P51449 1/20 0.31
PKM P14618 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.30
KLK7 P49862 1/20 0.30
CFTR P13569 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4566745 0.86 TSHR (0.32) HTT
SCHEMBL2414827 0.84 ALDH1A1 (0.33) ALDH1A1KDM4EKDM2BNR1H3HTT
SCHEMBL4566627 0.83 ABCC9 (0.33) KDM4ERORC
SCHEMBL2409056 0.82 KDM2B (0.35) ALDH1A1KDM4EKDM2BNR1H3HTT
SCHEMBL1580761 0.81 SLC40A1 (0.36) ALDH1A1KDM4EKDM2BHTTHSD11B1
SCHEMBL4566561 0.81 HTR6 (0.40) ALDH1A1RORC
Hydrochloric Acid SCHEMBL2415530 0.80 SLC40A1 (0.36) ALDH1A1KDM4EKDM2BHTTHSD11B1
SCHEMBL4566724 0.80
SCHEMBL2414830 0.80 PTGDR2 (0.34) ALDH1A1KDM4EKDM2BNR1H3HTT
Hydrochloric Acid SCHEMBL4422685 0.80 CFTR (0.30) CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed