SCHEMBL4566561

SCHEMBL4566561

CN(C(=O)OCc1cn(S(=O)(=O)c2ccc(OCc3ccccc3)cc2)c(-c2cccnc2F)c1F)C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.40
FFAR1 O14842 3/20 0.36
KEAP1 Q14145 1/20 0.35
MMP8 P22894 2/20 0.35
MMP3 P08254 1/20 0.35
AR P10275 2/20 0.35
NOX1 Q9Y5S8 1/20 0.35
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
MMP13 P45452 2/20 0.34
ADAMTS4 O75173 1/20 0.34
PTGES O14684 2/20 0.34
KCNH2 Q12809 2/20 0.34
ALOX5 P09917 1/20 0.33
RAB9A P51151 1/20 0.33
ALDH1A1 P00352 1/20 0.33
RORC P51449 1/20 0.33
MMP1 P03956 1/20 0.33
ADAM17 P78536 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2411207 0.85 HTR6 (0.39) HTR6FFAR1KEAP1MMP8MMP3
SCHEMBL4566599 0.85 RXFP1 (0.35) HTR6ALDH1A1
SCHEMBL4566627 0.85 ABCC9 (0.33) HTR6KEAP1RORC
SCHEMBL4422173 0.85 HTR6 (0.42) HTR6FFAR1KEAP1MMP8MMP3
SCHEMBL4566745 0.84 TSHR (0.32)
SCHEMBL2411210 0.83 HTR6 (0.38) HTR6FFAR1KEAP1MMP8MMP3
SCHEMBL2411204 0.81 ADAMTS4 (0.40) HTR6KEAP1MMP8ARMMP13
SCHEMBL4569945 0.81 ALDH1A1 (0.36) ALDH1A1RORC
SCHEMBL5002797 0.81 HTR6 (0.40) HTR6FFAR1KEAP1MMP8MMP3
SCHEMBL4566781 0.80

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed