SCHEMBL4568569

SCHEMBL4568569

Cc1ccc2c(Cc3cccc(C(=O)O)n3)c(-c3cccnc3)[nH]c2c1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MDM4 O15151 1/20 0.42
MDM2 Q00987 1/20 0.42
FNTA P49354 3/20 0.41
FNTB P49356 3/20 0.41
DHODH Q02127 2/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
ENPP2 Q13822 1/20 0.40
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
GPR35 Q9HC97 1/20 0.39
MAP2K4 P45985 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3701174 0.90 MDM4 (0.51) MDM4MDM2KDM4EENPP2
SCHEMBL4568492 0.90 MTNR1A (0.43) MDM4MDM2FNTAFNTBKDM4E
SCHEMBL3709676 0.89 KDM4E (0.43) FNTAFNTBDHODHKDM4ELMNA
SCHEMBL4568222 0.89 ENPP2 (0.45) FNTAFNTBENPP2
SCHEMBL3709862 0.88 KDM4E (0.52) KDM4EMTNR1AMTNR1BCYP11B1CYP11B2
SCHEMBL4568575 0.86 CYP19A1 (0.43) FNTAFNTBKDM4ELMNAMTNR1A
SCHEMBL4568573 0.86 ENPP2 (0.42) DHODHKDM4ELMNAHTTENPP2
SCHEMBL4568572 0.86 KDM4E (0.41) FNTAFNTBDHODHKDM4ELMNA
SCHEMBL4568571 0.86 DGAT1 (0.42) FNTAFNTBCYP11B1CYP11B2MAP2K4
SCHEMBL4568588 0.86 KDM4E (0.41) FNTAFNTBDHODHKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2474530-B1 INDOLE DERIVATIVE AND PHARMACOLOGICALLY ACCEPTABLE SALT THEREOF KISSEI PHARMACEUTICAL (JP) 2014-09-03 EP disclosed
US-20120122931-A1 INDOLE DERIVATIVE OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF KISSEI PHARMACEUTICAL CO., LTD. (JP) 2012-05-17 US disclosed
US-20120122931-A1 INDOLE DERIVATIVE OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF KISSEI PHARMACEUTICAL CO., LTD. (JP) 2012-05-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120122931-A1 INDOLE DERIVATIVE OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF PTGER1, CYSLTR1, LTB4R MDM4 4719/4885MDM2 2739/4885FNTA 1795/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.