SCHEMBL4570002

SCHEMBL4570002

COc1ccc(S(=O)(=O)n2cc(CCN(C(=O)O)C(C)(C)C)c(F)c2-c2cccnc2F)cn1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS2R14 Q9NYV8 1/20 0.33
NAMPT P43490 4/20 0.33
OXTR P30559 2/20 0.33
AVPR2 P30518 1/20 0.33
AVPR1A P37288 1/20 0.33
EIF2AK3 Q9NZJ5 1/20 0.32
MMP2 P08253 1/20 0.32
MMP9 P14780 1/20 0.32
MMP8 P22894 1/20 0.32
MMP13 P45452 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
KMT2A Q03164 1/20 0.32
RORC P51449 1/20 0.31
HTR6 P50406 6/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.30
HTR1A P08908 1/20 0.30
DRD2 P14416 1/20 0.30
HTR1D P28221 1/20 0.30
HTR1B P28222 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4570003 0.85 TAS2R14 (0.35) TAS2R14NAMPTOXTRAVPR2AVPR1A
SCHEMBL2409083 0.85 NAMPT (0.38) TAS2R14NAMPTOXTRAVPR2AVPR1A
SCHEMBL2409079 0.84 TAS2R14 (0.37) TAS2R14NAMPTOXTRAVPR2AVPR1A
SCHEMBL4570000 0.81 MMP2 (0.36) TAS2R14NAMPTOXTRAVPR2AVPR1A
SCHEMBL4570001 0.81 OXTR (0.34) TAS2R14NAMPTOXTRAVPR2AVPR1A
SCHEMBL1580223 0.81 EIF2AK3 (0.37) NAMPTOXTRAVPR2AVPR1AEIF2AK3
Fumaric Acid SCHEMBL2408204 0.80 NAMPT (0.37) TAS2R14NAMPTOXTRAVPR2AVPR1A
Fumaric Acid SCHEMBL2408214 0.80 NAMPT (0.37) TAS2R14NAMPTOXTRAVPR2AVPR1A
SCHEMBL17965497 0.80 NAMPT (0.36) TAS2R14NAMPTOXTRAVPR2AVPR1A
SCHEMBL1833794 0.76 PTGDR2 (0.34) MMP2MMP9MMP8MMP13PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed