SCHEMBL4570001

SCHEMBL4570001

COc1ccc(S(=O)(=O)n2cc(CN(C)C(=O)OC(C)(C)C)c(F)c2-c2cccnc2F)cn1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OXTR P30559 7/20 0.34
AVPR2 P30518 3/20 0.34
AVPR1A P37288 3/20 0.34
MMP2 P08253 2/20 0.33
MMP9 P14780 2/20 0.33
MMP8 P22894 2/20 0.33
MMP13 P45452 2/20 0.33
EIF2AK3 Q9NZJ5 1/20 0.33
NAMPT P43490 3/20 0.33
RORC P51449 1/20 0.33
TAS2R14 Q9NYV8 1/20 0.32
KAT6A Q92794 1/20 0.31
KAT5 Q92993 1/20 0.31
HTR2C P28335 1/20 0.30
SLC6A4 P31645 1/20 0.30
AAK1 Q2M2I8 1/20 0.30
ATM Q13315 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1833792 0.91 KAT6A (0.32) MMP2MMP9MMP8MMP13KAT6A
SCHEMBL2409079 0.89 TAS2R14 (0.37) OXTRAVPR2AVPR1AMMP2MMP9
SCHEMBL2411042 0.89 HTR6 (0.33) NAMPTRORCKAT6AKAT5HTR2C
SCHEMBL2409441 0.88 HTR2C (0.35) MMP2MMP9MMP8MMP13KAT6A
SCHEMBL2408854 0.87 NFE2L2 (0.34) OXTRMMP2MMP9MMP8MMP13
SCHEMBL2411540 0.86 MET (0.41) MMP2MMP9MMP8MMP13
SCHEMBL1278688 0.86 KAT6A (0.33) OXTRAVPR2AVPR1AMMP2MMP9
SCHEMBL2413759 0.85 RORC (0.36) NAMPTRORCKAT6AKAT5HTR2C
SCHEMBL1832149 0.85 HTR2C (0.33) NAMPTRORCKAT6AKAT5HTR2C
SCHEMBL4570003 0.85 TAS2R14 (0.35) OXTRAVPR2AVPR1AMMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed