SCHEMBL4573165

SCHEMBL4573165

O=S(=O)(CC1CC1)c1ccc(N2CCNCC2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.59
KDM4E B2RXH2 1/20 0.59
LMNA P02545 1/20 0.59
HTR6 P50406 4/20 0.56
ADRB1 P08588 5/20 0.47
SIRT6 Q8N6T7 1/20 0.47
HTR3E A5X5Y0 3/20 0.46
HTR3B O95264 3/20 0.46
HTR3A P46098 3/20 0.46
HTR3D Q70Z44 3/20 0.46
HTR3C Q8WXA8 3/20 0.46
SIGMAR1 Q99720 3/20 0.46
ADRB2 P07550 1/20 0.42
NCF1 P14598 1/20 0.42
PLD1 Q13393 1/20 0.42
USP2 O75604 1/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
MEN1 O00255 3/20 0.41
HRH4 Q9H3N8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5047347 0.79 SLC6A9 (0.42) ALDH1A1KDM4ELMNAHTR6CNR2
SCHEMBL10607953 0.78 ALDH1A1 (0.59) ALDH1A1KDM4ELMNAHTR6ADRB1
SCHEMBL9766413 0.77 ADRB1 (0.58) ALDH1A1KDM4ELMNAHTR6ADRB1
SCHEMBL31531621 0.76 ALDH1A1 (0.71) ALDH1A1KDM4ELMNAHTR6ADRB1
SCHEMBL4573220 0.76 ALDH1A1 (0.56) ALDH1A1KDM4ELMNAHTR6ADRB1
SCHEMBL532144 0.75 ALDH1A1 (0.69) ALDH1A1KDM4ELMNAHTR6ADRB1
SCHEMBL4518266 0.75 ALDH1A1 (1.00) ALDH1A1KDM4ELMNAHTR6ADRB1
SCHEMBL17968961 0.74 ADRB1 (0.49) ALDH1A1KDM4ELMNAADRB1SIRT6
SCHEMBL19485484 0.74 ADRB1 (0.49) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL17834368 0.74 ADRB1 (0.49) ALDH1A1KDM4ELMNAADRB1SIRT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed