SCHEMBL4573226

SCHEMBL4573226

COc1nc(N2CCNCC2)ccc1C1CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 5/20 0.47
HTR3E A5X5Y0 4/20 0.47
HTR3B O95264 4/20 0.47
HTR3A P46098 4/20 0.47
HTR3D Q70Z44 4/20 0.47
HTR3C Q8WXA8 4/20 0.47
HTR2C P28335 4/20 0.47
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
USP2 O75604 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
HTR1A P08908 1/20 0.47
MAPK1 P28482 1/20 0.47
SLC6A4 P31645 1/20 0.47
HTR7 P34969 1/20 0.47
HTT P42858 1/20 0.47
HTR6 P50406 1/20 0.47
PMP22 Q01453 1/20 0.47
HSD17B10 Q99714 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8117698 0.84 PRKCQ (0.41)
SCHEMBL26076035 0.79 HTR3E (0.51) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL4573932 0.79 UCHL3 (0.42) ALDH1A1KDM4EHSD17B10HRH3
SCHEMBL31651657 0.78 HTR3E (0.50) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL16422608 0.78 HTR3E (0.51) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL2875379 0.78 HTR3E (0.50) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL26074527 0.75 ADRB2 (0.49) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL26075869 0.75 HTR3E (0.48) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL5585294 0.74 ADRB2 (0.62) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL4573681 0.74 MAP4K4 (0.51) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed