SCHEMBL4573388

SCHEMBL4573388

CCOc1c(Cl)ccnc1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.40
LRRK2 Q5S007 1/20 0.38
HPGD P15428 2/20 0.37
KDM4E B2RXH2 2/20 0.37
GLA P06280 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
HSD17B10 Q99714 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CHUK O15111 1/20 0.36
GRM5 P41594 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
IKBKB O14920 2/20 0.35
NQO1 P15559 1/20 0.34
MAOA P21397 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9267937 0.79 MAOA (0.40) ALDH1A1MAPK1HTTHPGDKDM4E
SCHEMBL9261097 0.79 MAOA (0.40) ALDH1A1HPGDKDM4EGAAHSD17B10
SCHEMBL30230932 0.79 MAOA (0.48) ALDH1A1HPGDKDM4EHSD17B10L3MBTL1
SCHEMBL900450 0.79 MAOA (0.48) ALDH1A1HPGDKDM4EHSD17B10L3MBTL1
SCHEMBL19594501 0.79 GRM5 (0.47) ALDH1A1LRRK2HPGDKDM4EGLA
SCHEMBL9266335 0.78 PDE2A (0.36) ALDH1A1MAPK1HPGDKDM4EGAA
SCHEMBL9260347 0.78 SMN1; SMN2 (0.40) ALDH1A1MAPK1HTTHPGDKDM4E
SCHEMBL28136881 0.78 MAOA (0.42) ALDH1A1HTTHPGDKDM4EGAA
SCHEMBL9682836 0.77 LMNA (0.45) ALDH1A1MAPK1HTTHPGDKDM4E
SCHEMBL21061310 0.76 ALDH1A1 (0.39) ALDH1A1MAPK1LRRK2HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed
US-5877322-A Substituted pyridines, their preparation, and their use as pesticides and fungicides HOECHST SCHERING AGREVO GMBH (DE) 1999-03-02 US disclosed
US-5723450-A Substituted pyridines, their preparation, and their use as pesticides and fungicides HOECHST SCHERING AGREVO GMBH (DE) 1998-03-03 US disclosed
EP-0719256-A1 SUBSTITUTED PYRIDINES, PROCESS FOR PRODUCING THEM AND THEIR USE AS PESTICIDES AND FUNGICIDES Hoechst Schering AgrEvo GmbH (DE) 1996-07-03 EP disclosed
EP-0719257-A1 SUBSTITUTED PYRIDINES, PROCESS FOR PRODUCING THEM AND THEIR USE AS PESTICIDES AND FUNGICIDES Hoechst Schering AgrEvo GmbH (DE) 1996-07-03 EP disclosed
WO-1995007891-A1 SUBSTITUTED PYRIDINES, PROCESS FOR PRODUCING THEM AND THEIR USE AS PESTICIDES AND FUNGICIDES HOECHST SCHERING AGREVO GMBH (DE) 1995-03-23 WO disclosed
WO-1995007892-A1 SUBSTITUTED PYRIDINES, PROCESS FOR PRODUCING THEM AND THEIR USE AS PESTICIDES AND FUNGICIDES HOECHST SCHERING AGREVO GMBH (DE) 1995-03-23 WO disclosed