SCHEMBL4574178

SCHEMBL4574178

CC[C@H]1NC(=O)CN(Cc2cc(F)cc(F)c2F)C1=O

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 5/20 0.38
TACR1 P25103 1/20 0.35
RIPK1 Q13546 6/20 0.34
HDAC6 Q9UBN7 5/20 0.34
FNTA P49354 1/20 0.34
FNTB P49356 1/20 0.34
HDAC1 Q13547 4/20 0.33
HDAC8 Q9BY41 4/20 0.33
P2RX7 Q99572 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC7 Q8WUI4 1/20 0.31
HDAC10 Q969S8 1/20 0.31
HDAC11 Q96DB2 1/20 0.31
HDAC9 Q9UKV0 1/20 0.31
HDAC5 Q9UQL6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4574291 0.79 OPRK1 (0.46) OPRK1TACR1HDAC6FNTAFNTB
SCHEMBL3172734 0.76 OPRK1 (0.48) OPRK1TACR1HDAC6HDAC1HDAC8
SCHEMBL3172722 0.76 OPRK1 (0.48) OPRK1TACR1HDAC6HDAC1HDAC8
SCHEMBL4574124 0.72 RIPK1 (0.37) RIPK1FNTAFNTBP2RX7
SCHEMBL4574170 0.72 ATM (0.37) RIPK1FNTAFNTBP2RX7
SCHEMBL9836283 0.71 ALDH1A1 (0.39) OPRK1TACR1HDAC6HDAC1HDAC8
SCHEMBL334581 0.70 OPRK1 (0.59) OPRK1TACR1HDAC6HDAC1HDAC8
SCHEMBL6343378 0.70 OPRK1 (0.59) OPRK1TACR1HDAC6HDAC1HDAC8
SCHEMBL1714279 0.70 OPRK1 (0.59) OPRK1TACR1HDAC6HDAC1HDAC8
SCHEMBL14013787 0.69 RIPK1 (0.36) RIPK1FNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008134035-A1 ALPHA-UNSUBSTITUTED ARYLMETHYL PIPERAZINE PYRAZOLO[1,5-A] PYRIMIDINE AMIDE DERIVATIVES PANACOS PHARMACEUTICALS, INC. (US) 2008-11-06 WO disclosed
WO-2008134035-A1 ALPHA-UNSUBSTITUTED ARYLMETHYL PIPERAZINE PYRAZOLO[1,5-A] PYRIMIDINE AMIDE DERIVATIVES PANACOS PHARMACEUTICALS, INC. (US) 2008-11-06 WO disclosed