SCHEMBL4574291

SCHEMBL4574291

O=C1CN(Cc2cc(F)cc(F)c2F)C(=O)[C@@H](COCc2ccccc2)N1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 5/20 0.46
HDAC6 Q9UBN7 5/20 0.41
HDAC1 Q13547 4/20 0.40
HDAC8 Q9BY41 4/20 0.40
TACR1 P25103 1/20 0.40
FNTA P49354 1/20 0.38
FNTB P49356 1/20 0.38
ACKR3 P25106 1/20 0.38
HDAC4 P56524 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35
CYP3A4 P08684 1/20 0.35
TSHR P16473 1/20 0.35
LMNA P02545 1/20 0.34
AKT1 P31749 1/20 0.33
GRM5 P41594 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8574802 0.82 OPRK1 (0.56) OPRK1HDAC6HDAC1HDAC8TACR1
SCHEMBL8574805 0.82 OPRK1 (0.56) OPRK1HDAC6HDAC1HDAC8TACR1
SCHEMBL4574178 0.79 OPRK1 (0.38) OPRK1HDAC6HDAC1HDAC8TACR1
SCHEMBL6717771 0.74 OPRK1 (0.57) OPRK1HDAC6HDAC1HDAC8
SCHEMBL4293912 0.72 HDAC6 (0.60) OPRK1HDAC6HDAC1HDAC8TACR1
SCHEMBL3504268 0.71 GHSR (0.46) OPRK1CYP3A4TSHRLMNA
SCHEMBL3504617 0.71 GHSR (0.46) OPRK1CYP3A4TSHRLMNA
SCHEMBL3504265 0.71 GHSR (0.46) OPRK1CYP3A4TSHRLMNA
SCHEMBL4292380 0.70 OPRK1 (0.59) OPRK1HDAC6HDAC1HDAC8TACR1
SCHEMBL14033005 0.70 OPRK1 (0.61) OPRK1HDAC6HDAC1HDAC8TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008134035-A1 ALPHA-UNSUBSTITUTED ARYLMETHYL PIPERAZINE PYRAZOLO[1,5-A] PYRIMIDINE AMIDE DERIVATIVES PANACOS PHARMACEUTICALS, INC. (US) 2008-11-06 WO disclosed