SCHEMBL4574346

SCHEMBL4574346

Cc1nc2c3c(c(C(=O)N4CCC4)cn2c1C)CCC1(CCc2ccccc21)O3

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.34
AVPR1A P37288 5/20 0.33
LMNA P02545 3/20 0.33
TSHR P16473 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
SPR P35270 1/20 0.33
ALDH1A1 P00352 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
GLA P06280 1/20 0.33
HPGD P15428 1/20 0.33
RAB9A P51151 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PDK2 Q15119 1/20 0.32
AVPR2 P30518 1/20 0.32
NR1H2 P55055 2/20 0.32
NR1H3 Q13133 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596912 0.98 LMNA (0.35) HTTAVPR1ALMNATSHRNPSR1
SCHEMBL4595427 0.97 LMNA (0.35) HTTAVPR1ALMNATSHRNPSR1
SCHEMBL4575118 0.89 HCRTR1 (0.30) SPRHCRTR2
SCHEMBL4574395 0.89 HCAR2 (0.35) ALDH1A1RBP4
SCHEMBL4597065 0.89 HCRTR1 (0.33) LMNASMN1; SMN2HPGDHCRTR2
SCHEMBL4573882 0.85 SMN1; SMN2 (0.34) TSHRALDH1A1SMN1; SMN2KMT2AKDM4E
SCHEMBL4574534 0.77 CYP3A4 (0.31)
SCHEMBL14068675 0.77 ACACB (0.36) HTTAVPR1ALMNATSHRNPSR1
SCHEMBL4574391 0.76 MEN1 (0.30) KMT2AMEN1
SCHEMBL4738064 0.74 AVPR1A (0.34) AVPR1ALMNATSHRNPSR1SPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071766-A2 SPIRO-INDENE SUBSTITUTED IMIDAZONAPHYTHYRIDINE AND PYRANOIMIDAZOPYRIDINE DERIVATIVES AS INHIBITORS OF GASTRIC ACID SECRETION NYCOMED GMBH (DE) 2008-06-19 WO disclosed