SCHEMBL457788

SCHEMBL457788

CCc1[c]c(-c2ccc(Br)cc2)n[nH]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
IKBKB O14920 1/20 0.37
CHUK O15111 1/20 0.37
MEN1 O00255 1/20 0.35
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
KMT2A Q03164 1/20 0.35
PLCG1 P19174 1/20 0.34
MAPK1 P28482 2/20 0.33
MAPT P10636 2/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
METAP2 P50579 1/20 0.33
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL458788 0.82 BTK (0.36) NPC1RAB9ASMN1; SMN2ALDH1A1KMT2A
SCHEMBL455865 0.77 SMN1; SMN2 (0.46) NPC1RAB9ASMN1; SMN2IKBKBCHUK
SCHEMBL4637026 0.67 NR1H2 (0.40) NPC1RAB9ASMN1; SMN2MEN1USP2
SCHEMBL21198241 0.63 SMN1; SMN2 (0.66) NPC1RAB9ASMN1; SMN2MEN1USP2
SCHEMBL14790649 0.61 ERBB2 (0.50) NPC1RAB9ASMN1; SMN2IKBKBCHUK
SCHEMBL27519570 0.61 METAP2 (0.38) NPC1RAB9ASMN1; SMN2IKBKBCHUK
SCHEMBL20616131 0.60 HRH1 (0.46) NPC1RAB9ASMN1; SMN2MAPK1NFKB1
SCHEMBL2479806 0.60 MAPK1 (0.48) NPC1RAB9ASMN1; SMN2ALDH1A1MAPK1
Propane SCHEMBL27739979 0.59 CYP2A6 (0.67) SMN1; SMN2ALDH1A1PLCG1MAPK1GAA
SCHEMBL456840 0.58 IKBKB (0.43) IKBKBMETAP2NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614053-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2013-07-17 EP disclosed
WO-2012033225-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-03-15 WO disclosed