SCHEMBL4583237

SCHEMBL4583237

O=C(O)Nc1cc(-c2ccnc3c2ccn3S(=O)(=O)c2ccccc2)cs1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3C3 Q8NEB9 6/20 0.45
CYP2C19 P33261 1/20 0.45
HTR6 P50406 7/20 0.43
DRD2 P14416 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HTR2A P28223 1/20 0.37
RORC P51449 2/20 0.37
HDAC3 O15379 2/20 0.36
HDAC4 P56524 2/20 0.36
HDAC1 Q13547 2/20 0.36
HDAC7 Q8WUI4 2/20 0.36
HDAC2 Q92769 2/20 0.36
HDAC10 Q969S8 2/20 0.36
HDAC11 Q96DB2 2/20 0.36
HDAC8 Q9BY41 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36
HDAC9 Q9UKV0 2/20 0.36
HDAC5 Q9UQL6 2/20 0.36
ENPP3 O14638 1/20 0.36
ENPP1 P22413 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4584452 0.86 HTR6 (0.44) PIK3C3CYP2C19HTR6RORC
SCHEMBL10125133 0.85 L3MBTL1 (0.45) PIK3C3HTR6DRD2L3MBTL1RORC
SCHEMBL14510800 0.81 L3MBTL1 (0.41) PIK3C3L3MBTL1RORC
SCHEMBL4591926 0.80 AKT1 (0.43) PIK3C3CYP2C19HTR6L3MBTL1HDAC3
SCHEMBL4476225 0.80 L3MBTL1 (0.45) L3MBTL1RORC
SCHEMBL14494734 0.79 L3MBTL1 (0.44) PIK3C3CYP2C19HTR6L3MBTL1HDAC3
SCHEMBL8242143 0.79 PIK3C3 (0.39) PIK3C3CYP2C19HTR6RORC
SCHEMBL12346596 0.76 L3MBTL1 (0.43) PIK3C3CYP2C19HTR6L3MBTL1RORC
SCHEMBL8240222 0.75 RORC (0.42) PIK3C3CYP2C19HTR6RORC
SCHEMBL4593041 0.75 CYP2C19 (0.47) PIK3C3CYP2C19HTR6DRD2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968568-A2 INHIBITORS OF Akt ACTIVITY SmithKline Beecham Corporation (US) 2008-09-17 EP disclosed
WO-2007076423-A2 INHIBITORS OF Akt ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2007-07-05 WO disclosed