SCHEMBL4583470

SCHEMBL4583470

COc1ccc(C(N)C(NC(=O)O)C(C)(C)C)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.50
CNR2 P34972 1/20 0.43
RAB9A P51151 2/20 0.40
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
PAX8 Q06710 1/20 0.40
CNR1 P21554 3/20 0.40
KMT2A Q03164 2/20 0.40
ALDH1A1 P00352 2/20 0.40
TP53 P04637 1/20 0.40
CYP3A4 P08684 1/20 0.40
MEN1 O00255 1/20 0.40
ACACB O00763 1/20 0.40
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
GAA P10253 1/20 0.39
GPR88 Q9GZN0 1/20 0.39
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
PLK1 P53350 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4377187 0.83 DPP4 (0.43) MAPTKMT2AALDH1A1
SCHEMBL4373941 0.83 DPP4 (0.43) MAPTKMT2AALDH1A1
SCHEMBL4380602 0.82 PRCP (0.41) CNR2CNR1KMT2ACYP3A4MEN1
SCHEMBL4371626 0.82 ALDH1A1 (0.38) CNR2NPC1KMT2AALDH1A1CYP3A4
SCHEMBL3777012 0.74 LDHA (0.49) KMT2AALDH1A1ACACB
SCHEMBL1442862 0.74 GPR88 (0.48) NPSR1CNR2RAB9AKMT2AALDH1A1
SCHEMBL1673387 0.73 NPSR1 (0.47) NPSR1CNR2KMT2AALDH1A1CYP3A4
SCHEMBL6831820 0.73 LDHA (0.49) NPSR1RAB9ANPC1MAPTPAX8
SCHEMBL6046226 0.73 SLC1A3 (0.51) NPSR1RAB9ANPC1MAPTPAX8
SCHEMBL17334054 0.73 ACACB (0.62) NPSR1RAB9ACNR1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968568-A2 INHIBITORS OF Akt ACTIVITY SmithKline Beecham Corporation (US) 2008-09-17 EP disclosed
WO-2007076423-A2 INHIBITORS OF Akt ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2007-07-05 WO disclosed