SCHEMBL4585482

SCHEMBL4585482

Cc1cccc(Cl)c1C(=O)NC(C)CCN1CCC(N(Cc2cccc(C#N)c2)c2ccc(Oc3ccc(C(=O)O)cc3)cc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 17/20 0.51
KCNH2 Q12809 1/20 0.42
PGR P06401 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
DCUN1D1 Q96GG9 1/20 0.39
DRD2 P14416 1/20 0.38
DRD3 P35462 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4586226 0.91 CCR5 (0.50) CCR5KCNH2DCUN1D1DRD2DRD3
SCHEMBL4587594 0.89 CCR5 (0.48) CCR5KCNH2DCUN1D1DRD2DRD3
SCHEMBL4586220 0.86 CCR5 (0.43) CCR5KCNH2PGRCYP2D6CYP2C9
SCHEMBL4586072 0.86 CCR5 (0.57) CCR5KCNH2DCUN1D1DRD2DRD3
SCHEMBL4586809 0.86 CCR5 (0.50) CCR5KCNH2DCUN1D1DRD2DRD3
SCHEMBL4247926 0.86 CCR5 (0.70) CCR5
SCHEMBL4586727 0.86 CCR5 (0.51) CCR5KCNH2DCUN1D1
SCHEMBL4586981 0.84 CCR5 (0.49) CCR5KCNH2DCUN1D1DRD2DRD3
SCHEMBL4585280 0.83 CCR5 (0.48) CCR5PGRDCUN1D1DRD2DRD3
SCHEMBL4587080 0.83 CCR5 (0.51) CCR5KCNH2DCUN1D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed