SCHEMBL4586072

SCHEMBL4586072

Cc1cccc(C)c1C(=O)NC(C)CCN1CCC(N(Cc2ccccc2)c2ccc(Oc3ccc(C(=O)O)cc3)cc2)CC1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 9/20 0.57
DRD2 P14416 1/20 0.46
DRD3 P35462 1/20 0.46
LTA4H P09960 4/20 0.45
CACNA1B Q00975 1/20 0.44
KCNH2 Q12809 1/20 0.43
OPRM1 P35372 2/20 0.42
LPAR1 Q92633 2/20 0.41
LPAR5 Q9H1C0 2/20 0.41
UBE2M P61081 1/20 0.40
DCUN1D1 Q96GG9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4585297 0.93 CCR5 (0.48) CCR5DRD2DRD3CACNA1BKCNH2
SCHEMBL4586504 0.91 CCR5 (0.56) CCR5DRD2DRD3LTA4HCACNA1B
SCHEMBL4585280 0.87 CCR5 (0.48) CCR5DRD2DRD3UBE2MDCUN1D1
SCHEMBL4585572 0.87 CCR5 (0.52) CCR5DRD2DRD3CACNA1BKCNH2
SCHEMBL4585482 0.86 CCR5 (0.51) CCR5DRD2DRD3KCNH2DCUN1D1
SCHEMBL4586226 0.85 CCR5 (0.50) CCR5DRD2DRD3KCNH2DCUN1D1
SCHEMBL4586220 0.85 CCR5 (0.43) CCR5KCNH2
SCHEMBL4586422 0.85 CCR5 (0.47) CCR5DRD2DRD3UBE2MDCUN1D1
SCHEMBL4242440 0.82 CCR5 (0.81) CCR5
SCHEMBL4587594 0.82 CCR5 (0.48) CCR5DRD2DRD3CACNA1BKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed