SCHEMBL4585495

SCHEMBL4585495

COC(=O)c1cccc(N(Cc2cc(Cl)ccc2F)C2CCN(CCC(C)N)CC2)c1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PGR P06401 4/20 0.41
CYP2D6 P10635 4/20 0.41
CYP2C9 P11712 4/20 0.41
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41
OPRK1 P41145 1/20 0.41
CCR5 P51681 8/20 0.40
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
KCNH2 Q12809 1/20 0.39
HTR2A P28223 1/20 0.38
CASR P41180 1/20 0.37
UBE2M P61081 1/20 0.37
DCUN1D1 Q96GG9 1/20 0.37
SCN1A P35498 1/20 0.36
SCN8A Q9UQD0 1/20 0.36
BCHE P06276 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4586507 0.91 CCR5 (0.43) PGRCYP2D6CYP2C9CCR5NOS3
SCHEMBL4236571 0.86 CCR5 (0.48) PGRCYP2D6CYP2C9CCR5UBE2M
SCHEMBL4586676 0.84 CCR5 (0.40) PGRCYP2D6CYP2C9OPRM1OPRD1
SCHEMBL4586764 0.81 CCR5 (0.51) PGRCYP2D6CYP2C9OPRM1OPRD1
SCHEMBL4242919 0.81 MEN1 (0.51) PGRCYP2D6CYP2C9
SCHEMBL4586213 0.78 NOS3 (0.42) PGRCYP2D6CYP2C9CCR5NOS3
SCHEMBL4586037 0.77 PGR (0.42) PGRCYP2D6CYP2C9CCR5
SCHEMBL4236825 0.76 CCR5 (0.57) CCR5KCNH2
SCHEMBL4587113 0.76 CCR5 (0.57) PGRCYP2D6CYP2C9OPRM1OPRD1
SCHEMBL4242973 0.76 CCR5 (0.53) PGRCYP2D6CYP2C9CCR5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed