SCHEMBL4587113

SCHEMBL4587113

COC(=O)c1ccc(N(Cc2ccccc2)C2CCN(CCC(C)N)CC2)cc1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 8/20 0.57
DRD2 P14416 2/20 0.49
DRD3 P35462 1/20 0.49
UBE2M P61081 3/20 0.49
DCUN1D1 Q96GG9 3/20 0.49
OPRM1 P35372 3/20 0.46
OPRD1 P41143 1/20 0.46
OPRK1 P41145 1/20 0.46
HRH1 P35367 1/20 0.45
CACNA1B Q00975 1/20 0.45
PGR P06401 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4587621 0.97 CCR5 (0.55) CCR5DRD2DRD3UBE2MDCUN1D1
SCHEMBL4586715 0.96 CCR5 (0.55) CCR5DRD2DRD3UBE2MDCUN1D1
SCHEMBL4586764 0.90 CCR5 (0.51) CCR5DRD2DRD3UBE2MDCUN1D1
SCHEMBL4586343 0.88 CCR5 (0.51) CCR5DRD2DRD3DCUN1D1OPRM1
SCHEMBL4586731 0.85 OPRM1 (0.53) CCR5DRD2OPRM1CACNA1B
SCHEMBL4586689 0.84 CCR5 (0.51) CCR5DRD2DRD3DCUN1D1OPRM1
SCHEMBL4240429 0.83 CCR5 (0.68) CCR5UBE2MDCUN1D1
SCHEMBL4586507 0.82 CCR5 (0.43) CCR5PGRCYP2D6CYP2C9
SCHEMBL4585572 0.81 CCR5 (0.52) CCR5DRD2DRD3UBE2MDCUN1D1
SCHEMBL4586432 0.81 CCR5 (0.54) CCR5DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed