SCHEMBL4585644

SCHEMBL4585644

COC(=O)c1ccc(N(CC[C@@H](C)N)C2CCNCC2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.40
CCR5 P51681 2/20 0.39
EPHX1 P07099 1/20 0.38
OPRD1 P41143 1/20 0.37
LOXL2 Q9Y4K0 1/20 0.36
SLC6A4 P31645 5/20 0.36
SLC6A2 P23975 4/20 0.36
SLC6A3 Q01959 3/20 0.36
KCNH2 Q12809 3/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
GAA P10253 2/20 0.36
HPGD P15428 2/20 0.36
HSD17B10 Q99714 2/20 0.36
NPC1 O15118 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CACNA1B Q00975 2/20 0.36
MBTPS1 Q14703 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18361366 0.82 MEN1 (0.44) MAPTOPRD1LOXL2SLC6A4KCNH2
Hydrochloric Acid SCHEMBL21043567 0.81 MEN1 (0.44) MAPTOPRD1LOXL2SLC6A4KCNH2
SCHEMBL18361056 0.80 MEN1 (0.41) MAPTOPRD1LOXL2SLC6A4SLC6A2
Hydrochloric Acid SCHEMBL21043585 0.79 MEN1 (0.41) MAPTOPRD1LOXL2SLC6A4SLC6A2
SCHEMBL4585642 0.77 LOXL2 (0.39) MAPTEPHX1OPRD1LOXL2SLC6A4
SCHEMBL4247136 0.77 CCR5 (0.51) MAPTCCR5OPRD1SLC6A4SLC6A2
SCHEMBL4585576 0.75 HTR1F (0.36) GAACACNA1B
SCHEMBL18361035 0.75 NOTUM (0.46) MAPTOPRD1KDM4EALDH1A1GAA
SCHEMBL28363673 0.73 NOTUM (0.43) SLC6A4SLC6A2SLC6A3KCNH2KDM4E
SCHEMBL4587113 0.71 CCR5 (0.57) CCR5OPRD1CACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed