SCHEMBL4585780

SCHEMBL4585780

CC(C)(C)OC(=O)N1Cc2ccc(N(C(=O)OCc3ccccc3)C3CCNCC3)cc2C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 6/20 0.43
SIGMAR1 Q99720 6/20 0.43
HRH1 P35367 4/20 0.43
HRH3 Q9Y5N1 4/20 0.43
HRH2 P25021 3/20 0.43
HTR1A P08908 2/20 0.43
ADRA2C P18825 2/20 0.43
HTR2C P28335 2/20 0.43
ADRA2A P08913 1/20 0.43
ADRA2B P18089 1/20 0.43
DRD1 P21728 1/20 0.43
HTR1B P28222 1/20 0.43
HTR2A P28223 1/20 0.43
HTR1E P28566 1/20 0.43
SLC6A4 P31645 1/20 0.43
HTR2B P41595 1/20 0.43
ENPP2 Q13822 1/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
DDB1 Q16531 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17797540 0.72 ENPP2 (0.50) TMEM97SIGMAR1HRH1HRH3HTR1A
SCHEMBL12469312 0.71 SLC6A2 (0.46) SLC6A4MEN1KMT2ACHRM3SLC6A2
SCHEMBL4239069 0.70 ALDH1A1 (0.53) TMEM97SIGMAR1HRH1HRH3HRH2
SCHEMBL28699149 0.70 TMEM97 (0.77) TMEM97SIGMAR1HRH1HRH3HRH2
SCHEMBL30449380 0.70 TMEM97 (0.77) TMEM97SIGMAR1HRH1HRH3HRH2
SCHEMBL803663 0.70 JAK2 (0.54) SIGMAR1MEN1KMT2AJAK2JAK1
SCHEMBL2335192 0.70 HDAC1 (0.42) MEN1KMT2ADDB1CRBNHDAC1
SCHEMBL17560116 0.70 TACR1 (0.41) SLC6A4ENPP2MEN1KMT2ACHRM2
SCHEMBL21800218 0.70 TMEM97 (0.51) TMEM97SIGMAR1HRH1HRH3HRH2
SCHEMBL29593677 0.69 JAK2 (0.51) SIGMAR1MEN1KMT2AJAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed