SCHEMBL4586467

SCHEMBL4586467

CN(C)C(=O)C(C(N)=O)c1cc(Cl)c2[nH]c(=O)oc2c1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.35
GRM5 P41594 2/20 0.32
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.31
ADRA2A P08913 1/20 0.31
TSHR P16473 1/20 0.31
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
THPO P40225 1/20 0.31
BLM P54132 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5513581 0.72 KMO (0.37) KMOGRM5LMNACYP1A2ADRA2A
SCHEMBL5074233 0.71 KMO (0.39) KMOGRM5LMNACYP1A2ADRA2A
SCHEMBL5512753 0.71 KMO (0.39) KMOGRM5LMNACYP1A2ADRA2A
SCHEMBL14510182 0.68 KMO (0.36) KMOGRM5LMNACYP1A2ADRA2A
SCHEMBL5547929 0.68 NOS1 (0.49) KMOGRM5LMNACYP1A2ADRA2A
SCHEMBL4586262 0.68 KMO (0.31) KMO
SCHEMBL4585945 0.65 OPRK1 (0.32) GRM5
SCHEMBL7615467 0.65 ADRB2 (0.45) LMNACYP1A2TSHRBLM
SCHEMBL15319641 0.65 KMO (0.47) KMOGRM5LMNACYP1A2ADRA2A
SCHEMBL5547925 0.65 KMO (0.47) KMOGRM5LMNACYP1A2ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1689493-A4 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2008-04-23 EP claimed
EP-1689493-A1 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS Bristol-Myers Squibb Pharma Company (US) 2006-08-16 EP claimed
WO-2005065779-A1 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-07-21 WO claimed
EP-1539766-A1 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS Bristol-Myers Squibb Company (US) 2005-06-15 EP claimed
WO-2003104236-A1 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-12-18 WO claimed