SCHEMBL4586717

SCHEMBL4586717

COC(=O)c1ccc(N(Cc2cccc(Cl)c2)C2CCN(CCC(C)NC(=O)c3c(C)cccc3C)CC2)cc1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 15/20 0.50
PTGER4 P35408 1/20 0.43
DRD2 P14416 1/20 0.42
DRD3 P35462 1/20 0.42
PGR P06401 2/20 0.41
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41
OPRK1 P41145 1/20 0.41
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4585280 0.92 CCR5 (0.48) CCR5PTGER4DRD2DRD3PGR
SCHEMBL4585572 0.88 CCR5 (0.52) CCR5DRD2DRD3OPRM1OPRD1
SCHEMBL4586764 0.85 CCR5 (0.51) CCR5DRD2DRD3PGROPRM1
SCHEMBL4243348 0.83 CCR5 (0.72) CCR5
SCHEMBL4586756 0.82 CCR5 (0.62) CCR5PGRCYP2D6CYP2C9
SCHEMBL4585297 0.82 CCR5 (0.48) CCR5DRD2DRD3OPRM1
SCHEMBL4586072 0.81 CCR5 (0.57) CCR5DRD2DRD3OPRM1
SCHEMBL4586226 0.81 CCR5 (0.50) CCR5PTGER4DRD2DRD3
SCHEMBL4586088 0.79 CCR5 (0.42) CCR5DRD2DRD3PGRCYP2D6
SCHEMBL4586890 0.78 CCR5 (0.61) CCR5OPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed