SCHEMBL4585572

SCHEMBL4585572

COC(=O)c1ccc(Cc2ccc(N(Cc3ccccc3)C3CCN(CCC(C)NC(=O)c4c(C)cccc4C)CC3)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 12/20 0.52
DRD2 P14416 1/20 0.44
DRD3 P35462 1/20 0.44
KCNH2 Q12809 1/20 0.42
UBE2M P61081 1/20 0.42
DCUN1D1 Q96GG9 1/20 0.42
CACNA1B Q00975 1/20 0.40
HRH1 P35367 1/20 0.40
OPRM1 P35372 3/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4586717 0.88 CCR5 (0.50) CCR5DRD2DRD3OPRM1OPRD1
SCHEMBL4585297 0.87 CCR5 (0.48) CCR5DRD2DRD3KCNH2UBE2M
SCHEMBL4586072 0.87 CCR5 (0.57) CCR5DRD2DRD3KCNH2UBE2M
SCHEMBL4586715 0.85 CCR5 (0.55) CCR5DRD2DRD3UBE2MDCUN1D1
SCHEMBL4243466 0.83 CCR5 (0.75) CCR5UBE2MDCUN1D1
SCHEMBL4585280 0.82 CCR5 (0.48) CCR5DRD2DRD3UBE2MDCUN1D1
SCHEMBL4587113 0.81 CCR5 (0.57) CCR5DRD2DRD3UBE2MDCUN1D1
SCHEMBL4586226 0.80 CCR5 (0.50) CCR5DRD2DRD3KCNH2DCUN1D1
SCHEMBL4586422 0.79 CCR5 (0.47) CCR5DRD2DRD3UBE2MDCUN1D1
SCHEMBL4587621 0.79 CCR5 (0.55) CCR5DRD2DRD3UBE2MDCUN1D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed