SCHEMBL4587068

SCHEMBL4587068

CC(N)CCN1CCC(N(Cc2cccc(C#N)c2)c2ccc(OCC(=O)OC(C)(C)C)cc2)CC1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 13/20 0.48
KCNH2 Q12809 1/20 0.40
DCUN1D1 Q96GG9 1/20 0.39
MLNR O43193 1/20 0.39
CACNA1B Q00975 1/20 0.39
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38
SLC6A3 Q01959 2/20 0.38
MEN1 O00255 1/20 0.37
HTRA1 Q92743 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4586221 0.86 CCR5 (0.48) CCR5KCNH2DCUN1D1CACNA1BSLC6A2
SCHEMBL4242798 0.86 CCR5 (0.56) CCR5
SCHEMBL4240125 0.85 CCR5 (0.47) CCR5KCNH2CACNA1BSLC6A2SLC6A4
SCHEMBL4585533 0.84 CCR5 (0.50) CCR5KCNH2DCUN1D1MLNRSLC6A2
SCHEMBL4585633 0.83 CCR5 (0.47) CCR5KCNH2DCUN1D1SLC6A2SLC6A4
SCHEMBL4586343 0.83 CCR5 (0.51) CCR5KCNH2DCUN1D1
SCHEMBL4586689 0.83 CCR5 (0.51) CCR5KCNH2DCUN1D1CACNA1B
SCHEMBL4586071 0.80 KCNH2 (0.52) CCR5KCNH2DCUN1D1SLC6A2SLC6A4
SCHEMBL4241269 0.79 CCR5 (0.67) CCR5
SCHEMBL4586415 0.79 CCR5 (0.45) CCR5KCNH2DCUN1D1MLNRSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed