SCHEMBL4586071

SCHEMBL4586071

CC(N)CCN1CCC(N(Cc2cccc(C#N)c2)c2ccc([N+](=O)[O-])cc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.52
KCNJ1 P48048 2/20 0.52
CCR5 P51681 14/20 0.46
SLC6A2 P23975 2/20 0.40
SLC6A4 P31645 2/20 0.40
SLC6A3 Q01959 2/20 0.40
DCUN1D1 Q96GG9 1/20 0.39
PGR P06401 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4586335 0.87 CCR5 (0.53) CCR5DCUN1D1
SCHEMBL4586726 0.87 CCR5 (0.46) CCR5DCUN1D1PGR
SCHEMBL4586437 0.87 CCR5 (0.47) KCNH2KCNJ1CCR5DCUN1D1
SCHEMBL4586415 0.85 CCR5 (0.45) KCNH2CCR5SLC6A2SLC6A4SLC6A3
SCHEMBL4585533 0.85 CCR5 (0.50) KCNH2CCR5SLC6A2SLC6A4SLC6A3
SCHEMBL4586590 0.85 CCR5 (0.47) KCNH2CCR5SLC6A2SLC6A4SLC6A3
SCHEMBL4235948 0.84 CCR5 (0.55) KCNH2KCNJ1CCR5SLC6A2SLC6A4
SCHEMBL4586343 0.83 CCR5 (0.51) KCNH2CCR5DCUN1D1PGR
SCHEMBL4585633 0.83 CCR5 (0.47) KCNH2CCR5SLC6A2SLC6A4SLC6A3
SCHEMBL4587068 0.80 CCR5 (0.48) KCNH2CCR5SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed