SCHEMBL4586432

SCHEMBL4586432

CC(N)CCN1CCC(N(Cc2ccccc2)c2ccc(S(N)(=O)=O)cc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 6/20 0.54
CA12 O43570 12/20 0.51
CA1 P00915 12/20 0.51
CA2 P00918 12/20 0.51
CA4 P22748 12/20 0.51
CA5A P35218 12/20 0.51
CA7 P43166 12/20 0.51
CA9 Q16790 12/20 0.51
CA13 Q8N1Q1 12/20 0.51
CA14 Q9ULX7 12/20 0.51
DRD2 P14416 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4586335 0.85 CCR5 (0.53) CCR5DRD2
SCHEMBL4586731 0.83 OPRM1 (0.53) CCR5DRD2
SCHEMBL4236512 0.82 CCR5 (0.49) CCR5
SCHEMBL4587113 0.81 CCR5 (0.57) CCR5DRD2
SCHEMBL4587621 0.79 CCR5 (0.55) CCR5DRD2
SCHEMBL4586715 0.78 CCR5 (0.55) CCR5DRD2
SCHEMBL4586590 0.78 CCR5 (0.47) CCR5
SCHEMBL4586437 0.75 CCR5 (0.47) CCR5
SCHEMBL4586726 0.75 CCR5 (0.46) CCR5DRD2
SCHEMBL4585633 0.74 CCR5 (0.47) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed