SCHEMBL4587583

SCHEMBL4587583

CNC(=O)C(O)Cc1ccc(C(=O)O)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
ANPEP P15144 1/20 0.47
ENPEP Q07075 1/20 0.47
KMT2A Q03164 3/20 0.46
ADRB1 P08588 1/20 0.46
ADRB3 P13945 1/20 0.46
ACACB O00763 1/20 0.46
SRD5A2 P31213 1/20 0.45
FOLH1 Q04609 4/20 0.44
TDP1 Q9NUW8 2/20 0.43
TP53 P04637 1/20 0.41
TSHR P16473 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
USP2 O75604 1/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
THRB P10828 1/20 0.41
NR4A1 P22736 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25440208 0.84 NPC1 (0.50) KMT2ATSHRMEN1
SCHEMBL24988006 0.84 NPC1 (0.50) KMT2ATSHRMEN1
SCHEMBL3156555 0.84 NPC1 (0.50) KMT2ATSHRMEN1
SCHEMBL4587733 0.83 LOXL2 (0.53) KMT2ATDP1MEN1MAPT
SCHEMBL22857534 0.83 ACACB (0.49) ALDH1A1ANPEPENPEPKMT2AADRB1
SCHEMBL6243190 0.80 KDM6B (0.56) ALDH1A1ANPEPENPEPKMT2AADRB1
SCHEMBL7299745 0.79 MEN1 (0.51) ALDH1A1KMT2AMEN1SMN1; SMN2
SCHEMBL7300551 0.79 MEN1 (0.51) ALDH1A1KMT2AMEN1SMN1; SMN2
SCHEMBL28703199 0.79 MEN1 (0.51) ALDH1A1KMT2AMEN1SMN1; SMN2
SCHEMBL4598268 0.76 ALDH1A1 (0.57) ALDH1A1ANPEPENPEPKMT2AADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1973405-A2 HYDROXYALKYLARYLAMIDE DERIVATIVES Merck & Co., Inc. (US) 2008-10-01 EP disclosed
WO-2007087130-A2 HYDROXYALKYLARYLAMIDE DERIVATIVES MERCK & CO., INC. (US) 2007-08-02 WO disclosed