SCHEMBL4589447

SCHEMBL4589447

FC(F)(F)O[N]Cc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 5/20 0.42
TRPA1 O75762 2/20 0.39
ALDH1A1 P00352 2/20 0.39
CYP3A4 P08684 1/20 0.39
MIF P14174 1/20 0.39
HPGD P15428 1/20 0.39
CES1 P23141 1/20 0.36
TSHR P16473 3/20 0.36
GRIN1 Q05586 3/20 0.35
NOS2 P35228 1/20 0.35
CALM1 P0DP23 1/20 0.35
IDO1 P14902 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
EPHX2 P34913 1/20 0.33
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
GRIN2A Q12879 1/20 0.32
GRIN2C Q14957 1/20 0.32
GRIN3A Q8TCU5 1/20 0.32
SIGMAR1 Q99720 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6003245 0.83 GRIN2B (0.37) GRIN2BTRPA1ALDH1A1CYP3A4MIF
SCHEMBL5548041 0.70 ALDH1A1 (0.43) GRIN2BTRPA1ALDH1A1CYP3A4MIF
SCHEMBL8251 0.70 NOS2 (0.43) GRIN2BTRPA1ALDH1A1CYP3A4MIF
SCHEMBL7462793 0.70 TRPA1 (0.39) GRIN2BTRPA1ALDH1A1CYP3A4MIF
SCHEMBL4762887 0.68 TRPA1 (0.41) GRIN2BTRPA1ALDH1A1CYP3A4MIF
SCHEMBL6598540 0.68 TSHR (0.50) TRPA1ALDH1A1CYP3A4MIFHPGD
SCHEMBL1653 0.67 ALDH1A1 (0.55) GRIN2BTRPA1ALDH1A1CYP3A4MIF
SCHEMBL10667652 0.67 TSHR (0.44) GRIN2BTRPA1ALDH1A1CYP3A4MIF
SCHEMBL1852892 0.67 ALDH1A1 (0.40) GRIN2BTRPA1ALDH1A1CYP3A4MIF
SCHEMBL11337111 0.67 TP53 (0.44) GRIN2BTRPA1ALDH1A1CYP3A4MIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8329911-B2 Biphenyl compounds useful as muscarinic receptor antagonists THERAVANCE, INC. (US) 2012-12-11 US disclosed
WO-2008065500-A2 HETEROARYL AMIDES AS TYPE I GLYCINE TRANSPORT INHIBITORS PFIZER PRODUCTS INC. (US) 2008-06-05 WO disclosed
EP-0923562-B1 SUBSTITUTED P-TRIFLUOROMETHYLPHENYLURACILS BAYER AG (DE) 2002-10-09 EP disclosed
US-6444616-B1 HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2002-09-03 US disclosed
US-6130225-A Substituted p-trifluoromethylphenyluracils BAYER AKTIENGESELLSCHAFT (DE) 2000-10-10 US disclosed