SCHEMBL6003245

SCHEMBL6003245

FC(F)(F)C(F)(F)O[N]Cc1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 5/20 0.37
TRPA1 O75762 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 1/20 0.36
MIF P14174 1/20 0.36
HPGD P15428 1/20 0.36
CES1 P23141 2/20 0.34
GRIN1 Q05586 3/20 0.33
TSHR P16473 1/20 0.33
NOS2 P35228 1/20 0.33
CALM1 P0DP23 1/20 0.32
NR1H2 P55055 3/20 0.32
NR1H3 Q13133 3/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
EPHX2 P34913 1/20 0.31
IDO1 P14902 1/20 0.31
GRIN2D O15399 1/20 0.31
GRIN3B O60391 1/20 0.31
GRIN2A Q12879 1/20 0.31
GRIN2C Q14957 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4589447 0.83 GRIN2B (0.42) GRIN2BTRPA1ALDH1A1CYP3A4MIF
SCHEMBL5548041 0.67 ALDH1A1 (0.43) GRIN2BTRPA1ALDH1A1CYP3A4MIF
SCHEMBL8251 0.67 NOS2 (0.43) GRIN2BTRPA1ALDH1A1CYP3A4MIF
SCHEMBL7462793 0.67 TRPA1 (0.39) GRIN2BTRPA1ALDH1A1CYP3A4MIF
SCHEMBL6598540 0.66 TSHR (0.50) TRPA1ALDH1A1CYP3A4MIFHPGD
SCHEMBL4762887 0.66 TRPA1 (0.41) GRIN2BTRPA1ALDH1A1CYP3A4MIF
SCHEMBL28563732 0.65 CES1 (0.42) ALDH1A1HPGDCES1SMN1; SMN2IDO1
SCHEMBL1653 0.64 ALDH1A1 (0.55) GRIN2BTRPA1ALDH1A1CYP3A4MIF
SCHEMBL6003248 0.64 IDO1 (0.40) ALDH1A1CYP3A4HPGDCES1CALM1
SCHEMBL1852892 0.64 ALDH1A1 (0.40) GRIN2BTRPA1ALDH1A1CYP3A4MIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678185-A1 2,3-DIHYDRO-6-NITROIMIDAZO [2,1-B] OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-07-12 EP disclosed
WO-2005042542-A1 2,3-DIHYDRO-6-NITROIMIDAZO (2,1-B) OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2005-05-12 WO disclosed