SCHEMBL4589615

SCHEMBL4589615

FC(F)(F)c1cccc(C2CCN(CCc3ccc4cnccc4c3)CC2)n1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 13/20 0.49
DRD2 P14416 11/20 0.49
HTR1A P08908 10/20 0.49
KCNH2 Q12809 6/20 0.49
HRH3 Q9Y5N1 1/20 0.39
GRM2 Q14416 1/20 0.38
ROCK2 O75116 2/20 0.37
SLC6A4 P31645 2/20 0.37
CYP17A1 P05093 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A3 Q01959 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1401365 0.82 DRD2 (0.56) DRD4DRD2HTR1AGRM2ROCK2
Hydrochloric Acid SCHEMBL4589565 0.81 DRD2 (0.55) DRD4DRD2HTR1AGRM2ROCK2
SCHEMBL4589307 0.79 SIGMAR1 (0.50) DRD4DRD2HRH3ROCK2SLC6A4
SCHEMBL1401478 0.78 DRD2 (0.56) DRD4DRD2HTR1AGRM2ROCK2
SCHEMBL6589456 0.78 HTR1A (0.52) DRD4DRD2HTR1AKCNH2HRH3
SCHEMBL21662139 0.74 DRD4 (0.61) DRD4DRD2HTR1AKCNH2GRM2
SCHEMBL26446387 0.74 DRD2 (0.65) DRD4DRD2HTR1AKCNH2SLC6A4
SCHEMBL6586330 0.74 HTR1A (0.52) DRD4DRD2HTR1AKCNH2HRH3
Hydrochloric Acid SCHEMBL21642938 0.73 DRD4 (0.60) DRD4DRD2HTR1AKCNH2GRM2
SCHEMBL27460494 0.70 SIGMAR1 (0.39) DRD4DRD2KCNH2HRH3SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7326720-B2 Phenyl- and pyridylpiperidines with TNF activity SANOFI-AVENTIS (FR) 2008-02-05 US claimed