SCHEMBL4590232

SCHEMBL4590232

O=C(Cc1ccc2ncncc2c1)CC1CCN(Cc2ccccc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.52
DRD4 P21917 2/20 0.52
SIGMAR1 Q99720 1/20 0.47
ACHE P22303 3/20 0.44
BCHE P06276 2/20 0.44
GAA P10253 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3404965 0.86 DRD2 (0.56) DRD2DRD4SIGMAR1ACHE
SCHEMBL8819347 0.81 ACHE (0.54) DRD2DRD4SIGMAR1ACHEBCHE
SCHEMBL222191 0.79 ACHE (0.64) SIGMAR1ACHEBCHE
SCHEMBL4287273 0.79 DRD2 (0.50) DRD2DRD4SIGMAR1GAA
SCHEMBL7501904 0.79 DRD2 (0.63) DRD2DRD4SIGMAR1ACHEBCHE
SCHEMBL4289978 0.77 BCHE (0.69) DRD2DRD4SIGMAR1ACHEBCHE
Hydrochloric Acid SCHEMBL9381094 0.77 BCHE (0.69) DRD2DRD4SIGMAR1ACHEBCHE
SCHEMBL5259687 0.76 DRD2 (0.54) DRD2DRD4SIGMAR1GAA
SCHEMBL8818483 0.76 SIGMAR1 (0.64) DRD2DRD4SIGMAR1ACHE
SCHEMBL5039460 0.75 HRH3 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910384-A1 IMIDAZO [2,1-B]THIAYOLE DERIVATIVES AS SIRTUIN MODULATING COMPOUNDS Sirtris Pharmaceuticals, Inc. (US) 2008-04-16 EP disclosed
WO-2007019344-A1 IMIDAZO [2,1-B] THIAYOLE DERIVATIVES AS SIRTUIN MODULATING COMPOUNDS SIRTRIS PHARMACEUTICALS, INC. (US) 2007-02-15 WO disclosed
WO-2006094246-A2 N-ARYLMETHYL BENZAMIDE SIRTUIN MODULATORS SIRTRIS PHARMACEUTICALS, INC. (US) 2006-09-08 WO disclosed