SCHEMBL5259687

SCHEMBL5259687

O=C(Cc1ccc2occc2c1)CC1CCN(Cc2ccccc2)CC1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.54
DRD4 P21917 2/20 0.54
SIGMAR1 Q99720 3/20 0.49
FAAH O00519 1/20 0.45
GAA P10253 1/20 0.45
CXCR4 P61073 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7501904 0.81 DRD2 (0.63) DRD2DRD4SIGMAR1CXCR4
SCHEMBL4287273 0.79 DRD2 (0.50) DRD2DRD4SIGMAR1FAAHGAA
SCHEMBL8818483 0.79 SIGMAR1 (0.64) DRD2DRD4SIGMAR1FAAH
SCHEMBL3404965 0.78 DRD2 (0.56) DRD2DRD4SIGMAR1
SCHEMBL220604 0.78 ACHE (0.66) SIGMAR1
SCHEMBL4590232 0.76 DRD2 (0.52) DRD2DRD4SIGMAR1GAA
SCHEMBL4289978 0.76 BCHE (0.69) DRD2DRD4SIGMAR1
Hydrochloric Acid SCHEMBL9381094 0.75 BCHE (0.69) DRD2DRD4SIGMAR1
SCHEMBL4284929 0.74 DRD2 (0.59) DRD2DRD4FAAHCXCR4
SCHEMBL6262731 0.73 ACHE (0.68) DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1853610-A1 N-PHENYL BENZAMIDE DERIVATIVES AS SIRTUIN MODULATORS Sirtris Pharmaceuticals, Inc. (US) 2007-11-14 EP disclosed
EP-1850840-A2 NOVEL COMPOSITIONS FOR PREVENTING AND TREATING NEURODEGENERATIVE AND BLOOD COAGULATION DISORDERS Sirtris Pharmaceuticals, Inc. (US) 2007-11-07 EP disclosed
WO-2006094236-A1 N-PHENYL BENZAMIDE DERIVATIVES AS SIRTUIN MODULATORS SIRTRIS PHARMACEUTICALS, INC. (US) 2006-09-08 WO disclosed
WO-2006094209-A2 N-BENZIMIDAZOLYLALKYL-SUBSTITUTED AMIDE SIRTUIN MODULATORS SIRTRIS PHARMACEUTICALS, INC. (US) 2006-09-08 WO disclosed
WO-2006094248-A1 ARYL-SUBSTITUTED CYCLIC SIRTUIN MODULATORS SIRTRIS PHARMACEUTICALS, INC. (US) 2006-09-08 WO disclosed
WO-2006078941-A2 NOVEL SIRTUIN ACTIVATING COMPOUNDS AND METHODS OF USE THEREOF SIRTRIS PHARMACEUTICALS, INC. (US) 2006-07-27 WO disclosed
WO-2006076681-A2 NOVEL COMPOSITIONS FOR PREVENTING AND TREATING NEURODEGENERATIVE AND BLOOD COAGULATION DISORDERS SIRTRIS PHARMACEUTICALS, INC. (US) 2006-07-20 WO disclosed