SCHEMBL4590891

SCHEMBL4590891

C[C@@H]1CN(Cc2cc(F)cc(F)c2F)[C@@H](C)CN1

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.43
RIPK1 Q13546 3/20 0.38
XIAP P98170 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31305862 0.83 SIGMAR1 (0.49) SIGMAR1XIAP
SCHEMBL4574098 0.78 RIPK1 (0.38) RIPK1
SCHEMBL4575085 0.78 RIPK1 (0.38) RIPK1
SCHEMBL14566377 0.77 SIGMAR1 (0.51) SIGMAR1XIAP
SCHEMBL2022959 0.76 XIAP (0.40) XIAP
SCHEMBL31305848 0.76 SIGMAR1 (0.42) SIGMAR1XIAP
SCHEMBL4678046 0.74 SIGMAR1 (0.56) SIGMAR1
SCHEMBL4590115 0.74 SIGMAR1 (0.40) SIGMAR1RIPK1
SCHEMBL5058871 0.74 SIGMAR1 (0.56) SIGMAR1
SCHEMBL3165725 0.74 SIGMAR1 (0.56) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008134035-A1 ALPHA-UNSUBSTITUTED ARYLMETHYL PIPERAZINE PYRAZOLO[1,5-A] PYRIMIDINE AMIDE DERIVATIVES PANACOS PHARMACEUTICALS, INC. (US) 2008-11-06 WO disclosed
WO-2008134035-A1 ALPHA-UNSUBSTITUTED ARYLMETHYL PIPERAZINE PYRAZOLO[1,5-A] PYRIMIDINE AMIDE DERIVATIVES PANACOS PHARMACEUTICALS, INC. (US) 2008-11-06 WO disclosed