SCHEMBL4574098

SCHEMBL4574098

C[C@H]1CNCCN1Cc1cc(F)cc(F)c1F

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 3/20 0.38
HTR2C P28335 5/20 0.35
HTR2A P28223 4/20 0.35
HTR2B P41595 4/20 0.35
DPP4 P27487 1/20 0.34
KCNH2 Q12809 1/20 0.33
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4575085 1.00 RIPK1 (0.38) RIPK1HTR2CHTR2AHTR2BDPP4
SCHEMBL4590891 0.78 SIGMAR1 (0.43) RIPK1
SCHEMBL4574455 0.74 KDM4E (0.44) KCNH2CYP1A2KMT2A
SCHEMBL29050285 0.74 ALDH1A1 (0.44) KCNH2KMT2A
SCHEMBL4574384 0.71 RIPK1 (0.43) RIPK1DPP4
SCHEMBL4591030 0.71 RIPK1 (0.43) RIPK1DPP4
SCHEMBL4591026 0.71 RIPK1 (0.43) RIPK1DPP4
SCHEMBL2022959 0.70 XIAP (0.40) CYP3A4
SCHEMBL20818079 0.70 LMNA (0.56) HTR2CDPP4KCNH2KMT2A
SCHEMBL26192287 0.69 ALDH1A1 (0.54) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008134035-A1 ALPHA-UNSUBSTITUTED ARYLMETHYL PIPERAZINE PYRAZOLO[1,5-A] PYRIMIDINE AMIDE DERIVATIVES PANACOS PHARMACEUTICALS, INC. (US) 2008-11-06 WO disclosed
WO-2008134035-A1 ALPHA-UNSUBSTITUTED ARYLMETHYL PIPERAZINE PYRAZOLO[1,5-A] PYRIMIDINE AMIDE DERIVATIVES PANACOS PHARMACEUTICALS, INC. (US) 2008-11-06 WO disclosed